SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats (Q24672651)

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Sergio Melotto

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Mario Massagrande

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Andrew D Gribble

4

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Phillip Jeffrey

5

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Alexander J Stevens

6

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Nigel J Deeks

7

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Peter J Eddershaw

8

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Susan H Fenwick

9

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Graham Riley

10

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Tania Stean

11

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Claire M Scott

12

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Derek N Middlemiss

14

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Jim J Hagan

15

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Gary W Price

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Ian T Forbes

full work available at URL

17

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language of work or name

English

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publication date

June 2003

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https://www.ncbi.nlm.nih.gov/pmc/articles/PMC1573887

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published in

British Journal of Pharmacology

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volume

139

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issue

4

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page(s)

705-14

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cites work

Characterization of [(125)I]-SB-258585 binding to human recombinant and native 5-HT(6) receptors in rat, pig and human brain tissue

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5-CT stimulation of adenylyl cyclase activity in guinea-pig hippocampus: evidence for involvement of 5-HT7 and 5-HT1A receptors

7 April 2017

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Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase

7 April 2017

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

7 April 2017

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A novel adenylyl cyclase-activating serotonin receptor (5-HT7) implicated in the regulation of mammalian circadian rhythms

7 April 2017

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[(3)H]-SB-269970--A selective antagonist radioligand for 5-HT(7) receptors

7 April 2017

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Functional characterisation of the human cloned 5-HT7 receptor (long form); antagonist profile of SB-258719

7 April 2017

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Some quantitative uses of drug antagonists

7 April 2017

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SB-656104-A: a novel 5-HT(7) receptor antagonist with improved in vivo properties

7 April 2017

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The neurobiology of sleep: genetics, cellular physiology and subcortical networks

28 September 2017

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Localization of 5-HT(7) receptors in rat brain by immunocytochemistry, in situ hybridization, and agonist stimulated cFos expression.

28 September 2017

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Depression and sleep disorders: clinical relevance, economic burden and pharmacological treatment

28 September 2017

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Characterization of SB-269970-A, a selective 5-HT(7) receptor antagonist

28 September 2017

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A novel, potent, and selective 5-HT(7) antagonist: (R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolidine-1-sulfonyl) phen ol (SB-269970).

28 September 2017

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Function and distribution of three rat 5-hydroxytryptamine7 (5-HT7) receptor isoforms produced by alternative splicing

28 September 2017

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Contribution of the circadian pacemaker and the sleep homeostat to sleep propensity, sleep structure, electroencephalographic slow waves, and sleep spindle activity in humans.

28 September 2017

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Characterization and distribution of putative 5-ht7 receptors in guinea-pig brain

28 September 2017

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Cloning and expression of a 5-hydroxytryptamine7 receptor positively coupled to adenylyl cyclase

28 September 2017

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Pharmacological studies with SK&F 93944 (temelastine), a novel histamine H1-receptor antagonist with negligible ability to penetrate the central nervous system

28 September 2017

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Neural regulation of circadian rhythms

28 September 2017

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Evidence that wakefulness and REM sleep are controlled by a GABAergic pontine mechanism

28 September 2017

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Effects of antidepressants on 5-HT7 receptor regulation in the rat hypothalamus

30 May 2018

1 reference

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Inhibition by 5-HT7 receptor stimulation of GABAA receptor-activated current in cultured rat suprachiasmatic neurones

30 May 2018

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https://api.crossref.org/works/10.1038%2FSJ.BJP.0705290

Effect of bupropion-SR on REM sleep: relationship to antidepressant response

21 January 2018

1 reference

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DR4004, a putative 5-HT(7) receptor antagonist, also has functional activity at the dopamine D2 receptor.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1573887

5-HT7 receptors modulate synchronized network activity in rat hippocampus

28 November 2018

1 reference

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[3H]-SB-269970 radiolabels 5-HT7 receptors in rodent, pig and primate brain tissues

28 November 2018

1 reference

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In vivo resetting of the hamster circadian clock by 5-HT7 receptors in the suprachiasmatic nucleus.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1573887

A 5-HT(7) receptor-mediated depolarization in the anterodorsal thalamus. I. Pharmacological characterization.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1573887

Circadian variation of EEG power spectra in NREM and REM sleep in humans: dissociation from body temperature

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1573887

5-HT7 receptors mediate serotonergic effects on light-sensitive suprachiasmatic nucleus neurons

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1573887

Pharmacological characterisation of [35S]-GTPgammaS binding to Chinese hamster ovary cell membranes stably expressing cloned human 5-HT1D receptor subtypes

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1573887

5-Hydroxytryptamine(7) receptor activation decreases slow afterhyperpolarization amplitude in CA3 hippocampal pyramidal cells

28 November 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/12812993

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/12812993

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identification of 5-hydroxytryptamine7 receptor binding sites in rat hypothalamus: sensitivity to chronic antidepressant treatment

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/12812993