Binding of an octylglucoside detergent molecule in the second substrate (S2) site of LeuT establishes an inhibitor-bound conformation (Q27654242)

4

0 references

Anne-Marie Lund Winther

Anne-Marie Lund Winther

2

0 references

Jonathan Javitch

Jonathan A Javitch

6

0 references

Lei Shi

Lei Shi

3

0 references

Harel Weinstein

Harel Weinstein

5

0 references

author name string

Matthias Quick

Proceedings of the National Academy of Sciences of the United States of America

1

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language of work or name

English

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publication date

7 April 2009

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published in

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volume

106

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issue

14

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page(s)

5563-8

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cites work

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LeuT-desipramine structure reveals how antidepressants block neurotransmitter reuptake

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Antidepressant binding site in a bacterial homologue of neurotransmitter transporters

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Allelic heterogeneity at the serotonin transporter locus (SLC6A4) confers susceptibility to autism and rigid-compulsive behaviors

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Plasma membrane monoamine transporters: structure, regulation and function

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All-atom empirical potential for molecular modeling and dynamics studies of proteins

20 March 2017

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Phasercrystallographic software

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Scalable molecular dynamics with NAMD

20 March 2017

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Coot: model-building tools for molecular graphics

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PHENIX: building new software for automated crystallographic structure determination

20 March 2017

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20 March 2017

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Crystal structure of a bacterial homologue of Na+/Cl--dependent neurotransmitter transporters

22 April 2017

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A rapid, sensitive, and specific method for the determination of protein in dilute solution

7 April 2017

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Recent developments in the design of anti-depressive therapies: targeting the serotonin transporter

7 April 2017

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29 September 2017

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Monitoring the function of membrane transport proteins in detergent-solubilized form

29 September 2017

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Enhancement of drug absorption by noncharged detergents through membrane and P-glycoprotein binding

29 September 2017

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How did the neurotransmitter cross the bilayer? A closer view

29 September 2017

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Role of the GABA transporter in epilepsy.

29 September 2017

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Monoamine transporters and psychostimulant drugs

29 September 2017

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Serotonin transporter missense mutation associated with a complex neuropsychiatric phenotype

29 September 2017

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29 September 2017

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Stable expression of biogenic amine transporters reveals differences in inhibitor sensitivity, kinetics, and ion dependence.

29 September 2017

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Neurotransmitter transporters as molecular targets for addictive drugs.

2 June 2018

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Increased serotonin transporter availability in the brainstem of migraineurs

21 January 2018

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The mechanism of a neurotransmitter:sodium symporter--inward release of Na+ and substrate is triggered by substrate in a second binding site

21 January 2018

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The uncoupled chloride conductance of a bacterial glutamate transporter homolog

21 January 2018

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Carbohydrate solution simulations: producing a force field with experimentally consistent primary alcohol rotational frequencies and populations

21 January 2018

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Identification and selective inhibition of the channel mode of the neuronal GABA transporter 1.

21 January 2018

1 reference

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Interactions of alkylglucosides with the renal sodium/D-glucose cotransporter

27 November 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19307590

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.0811322106

1 reference

ADS bibcode

2009PNAS..106.5563Q

0 references

1 reference

1 reference

PubMed publication ID

19307590

1 reference