[Nphe1,Arg14,Lys15]nociceptin-NH2, a novel potent and selective antagonist of the nociceptin/orphanin FQ receptor. (Q35044357)

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8 November 2019

title

[Nphe1,Arg14,Lys15]nociceptin-NH2, a novel potent and selective antagonist of the nociceptin/orphanin FQ receptor (English)

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8 November 2019

0 references

7

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8 November 2019

David G Lambert

10

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8 November 2019

12

Domenico Regoli

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8 November 2019

1

Girolamo Calo

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8 November 2019

author name string

Anna Rizzi

2

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8 November 2019

Daniela Rizzi

3

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8 November 2019

Raffaella Bigoni

4

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8 November 2019

Remo Guerrini

5

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8 November 2019

Giuliano Marzola

6

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8 November 2019

John McDonald

8

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8 November 2019

Michele Morari

9

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8 November 2019

Severo Salvadori

11

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8 November 2019

language of work or name

English

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publication date

1 May 2002

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British Journal of Pharmacology

8 November 2019

published in

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8 November 2019

volume

136

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8 November 2019

issue

2

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8 November 2019

page(s)

303-311

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The molecular and behavioral pharmacology of the orphanin FQ/nociceptin peptide and receptor family

8 November 2019

cites work

1 reference

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Characterization of the locomotor activity-inhibiting effect of nociceptin/orphanin FQ in mice.

8 July 2018

1 reference

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Retro-nociceptin methylester, a peptide with analgesic and memory-enhancing activity.

8 July 2018

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4-Aminoquinolines: novel nociceptin antagonists with analgesic activity

8 July 2018

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Highly potent nociceptin analog containing the Arg-Lys triple repeat

8 July 2018

1 reference

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Nociceptin/orphanin FQ receptor ligands.

8 July 2018

1 reference

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In vitro and in vivo pharmacological characterization of J-113397, a potent and selective non-peptidyl ORL1 receptor antagonist

8 July 2018

1 reference

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Pharmacology of nociceptin and its receptor: a novel therapeutic target

8 July 2018

1 reference

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Characterization of [Nphe(1)]nociceptin(1-13)NH(2), a new selective nociceptin receptor antagonist

8 July 2018

1 reference

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Ligands for kappa-opioid and ORL1 receptors identified from a conformationally constrained peptide combinatorial library

8 July 2018

1 reference

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Comparison of the effects of [Phe1psi(CH2-NH)Gly2]nociceptin(1-13)NH2 in rat brain, rat vas deferens and CHO cells expressing recombinant human nociceptin receptors

8 July 2018

1 reference

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Loss of antinociception induced by naloxone benzoylhydrazone in nociceptin receptor-knockout mice.

8 July 2018

1 reference

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Effects of C-terminal truncation of the recombinant delta-opioid receptor on phospholipase C and adenylyl cyclase coupling.

8 July 2018

1 reference

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Address and message sequences for the nociceptin receptor: a structure-activity study of nociceptin-(1-13)-peptide amide.

8 July 2018

1 reference

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Unrestrained nociceptive response and disregulation of hearing ability in mice lacking the nociceptin/orphaninFQ receptor

8 July 2018

1 reference

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The effects of recombinant rat mu-opioid receptor activation in CHO cells on phospholipase C, [Ca2+]i and adenylyl cyclase.

8 July 2018

1 reference

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International Union of Pharmacology Committee on Receptor Nomenclature and Drug Classification. IX. Recommendations on terms and symbols in quantitative pharmacology.

8 July 2018

1 reference

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Isolation and structure of the endogenous agonist of opioid receptor-like ORL1 receptor

8 July 2018

1 reference

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Guanine nucleotide-binding protein-coupled and -uncoupled states of opioid receptors and their relevance to the determination of subtypes

8 July 2018

1 reference

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Characterisation of the non-peptide nociceptin receptor agonist, Ro64-6198 in Chinese hamster ovary cells expressing recombinant human nociceptin receptors

8 July 2018

1 reference

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[Arg(14),Lys(15)]nociceptin, a highly potent agonist of the nociceptin/orphanin FQ receptor: in vitro and in vivo studies

25 October 2018

1 reference

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Studies on the antinociceptive effect of [Nphe1]nociceptin(1-13)NH2 in mice

25 October 2018

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[Nphe(1)]NC(1-13)NH(2) selectively antagonizes nociceptin/orphanin FQ-stimulated G-protein activation in rat brain.

25 October 2018

1 reference

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Modulation of 5-hydroxytryptamine efflux from rat cortical synaptosomes by opioids and nociceptin

25 October 2018

1 reference

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[Nphe(1)]nociceptin-(1-13)-NH(2) antagonizes nociceptin effects in the mouse colon.

25 October 2018

1 reference

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Characterization of nociceptin receptors in the periphery: in vitro and in vivo studies

25 October 2018

1 reference

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NMDA and non-NMDA ionotropic glutamate receptors modulate striatal acetylcholine release via pre- and postsynaptic mechanisms

25 October 2018

1 reference

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Pharmacological characterization of the nociceptin receptor mediating hyperalgesia in the mouse tail withdrawal assay

25 October 2018

1 reference

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Orphanin FQ: a neuropeptide that activates an opioidlike G protein-coupled receptor.

25 October 2018

1 reference

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In vitro characterization of J-113397, a non-peptide nociceptin/orphanin FQ receptor antagonist

25 October 2018

1 reference

12 December 2020

Further Studies on Nociceptin-Related Peptides: Discovery of a New Chemical Template with Antagonist Activity on the Nociceptin Receptor

1 reference

12 December 2020

Intracerebroventricular injections in mice. Some methodological refinements

1 reference

12 December 2020

Association of aminopeptidase N and endopeptidase 24.15 inhibitors potentiate behavioral effects mediated by nociceptin/orphanin FQ in mice

1 reference

12 December 2020

Structure–activity studies on nociceptin/orphanin FQ: from full agonist, to partial agonist, to pure antagonist

1 reference

12 December 2020

Identifiers

DOI

10.1038/SJ.BJP.0704706

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12010780%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12010780%20AND%20SRC:MED&resulttype=core&format=json

8 November 2019

PubMed publication ID

12010780

1 reference