Binding ensemble profiling with photoaffinity labeling (BEProFL) approach: mapping the binding poses of HDAC8 inhibitors (Q37463122)

20 August 2017

Binding ensemble profiling with photoaffinity labeling (BEProFL) approach: mapping the binding poses of HDAC8 inhibitors (English)

1 reference

20 August 2017

8

Richard van Breemen

1 reference

20 August 2017

Bai He

1

1 reference

20 August 2017

Subash Velaparthi

2

1 reference

20 August 2017

Gilles Pieffet

3

1 reference

20 August 2017

Chris Pennington

4

1 reference

20 August 2017

Aruna Mahesh

5

1 reference

20 August 2017

Denise L Holzle

6

1 reference

20 August 2017

Michael Brunsteiner

7

1 reference

20 August 2017

Sylvie Y Blond

9

1 reference

20 August 2017

Pavel A Petukhov

10

1 reference

20 August 2017

language of work or name

English

0 references

publication date

1 November 2009

1 reference

Journal of Medicinal Chemistry

20 August 2017

1 reference

20 August 2017

52

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20 August 2017

22

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20 August 2017

7003-7013

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describes a project that uses

20 August 2017

ImageJ

1 reference

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC2789734/fullTextXML

inferred from PubMed Central ID database lookup

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Structural Studies of Human Histone Deacetylase 8 and Its Site-Specific Variants Complexed with Substrate and Inhibitors † , ‡

23 August 2017

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Histone deacetylase inhibitors: a novel class of anti-cancer agents on its way to the market

23 August 2017

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Histone deacetylase inhibitors: possible implications for neurodegenerative disorders

23 August 2017

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Substrate binding to histone deacetylases as shown by the crystal structure of the HDAC8-substrate complex

23 August 2017

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23 August 2017

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Activity-based probes for proteomic profiling of histone deacetylase complexes

23 August 2017

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23 August 2017

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23 August 2017

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23 August 2017

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Does water play a structural role in the folding of small nucleic acids?

23 August 2017

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23 August 2017

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23 August 2017

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Affordable image analysis using NIH Image/ImageJ

23 August 2017

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A chemical approach for identifying O-GlcNAc-modified proteins in cells

23 August 2017

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Histone deacetylases (HDACs): characterization of the classical HDAC family

23 August 2017

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Fast, efficient generation of high-quality atomic charges. AM1-BCC model: II. Parameterization and validation

23 August 2017

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Incorporation of azides into recombinant proteins for chemoselective modification by the Staudinger ligation

23 August 2017

1 reference

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Histone deacetylase inhibitors: inducers of differentiation or apoptosis of transformed cells

23 August 2017

1 reference

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Cell surface engineering by a modified Staudinger reaction

23 August 2017

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Development and validation of a genetic algorithm for flexible docking

23 August 2017

1 reference

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

23 August 2017

1 reference

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A series of potent and selective, triazolylphenyl-based histone deacetylases inhibitors with activity against pancreatic cancer cells and Plasmodium falciparum

23 August 2017

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A tandem orthogonal proteolysis strategy for high-content chemical proteomics

14 September 2017

1 reference

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A "traceless" Staudinger ligation for the chemoselective synthesis of amide bonds

26 June 2018

1 reference

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A functional proteomic strategy to discover inhibitors for uncharacterized hydrolases

26 June 2018

1 reference

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Functional differences in epigenetic modulators-superiority of mercaptoacetamide-based histone deacetylase inhibitors relative to hydroxamates in cortical neuron neuroprotection studies

2 September 2018

1 reference

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Synthesis of a bis-azido analogue of acromelic acid for radioisotope-free photoaffinity labeling and biochemical studies

2 September 2018

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Design of dantrolene-derived probes for radioisotope-free photoaffinity labeling of proteins involved in the physiological Ca2+ release from sarcoplasmic reticulum of skeletal muscle.

2 September 2018

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Microarray platform for profiling enzyme activities in complex proteomes

2 September 2018

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A strategy for functional proteomic analysis of glycosidase activity from cell lysates.

2 September 2018

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Structural snapshots of human HDAC8 provide insights into the class I histone deacetylases

2 September 2018

1 reference

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Thiol-based SAHA analogues as potent histone deacetylase inhibitors

2 September 2018

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Novel bifunctional probe for radioisotope-free photoaffinity labeling: compact structure comprised of photospecific ligand ligation and detectable tag anchoring units

2 September 2018

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Mapping enzyme active sites in complex proteomes

2 September 2018

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Activity-based protein profiling in vivo using a copper(i)-catalyzed azide-alkyne [3 + 2] cycloaddition

2 September 2018

1 reference

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Investigating cellular metabolism of synthetic azidosugars with the Staudinger ligation

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789734

Orientation of GTP and ADP within their respective binding sites in glutamate dehydrogenase

2 September 2018

1 reference

12 December 2020

Photoaffinity labeling of creatine kinase with 2-azido- and 8-azidoadenosine triphosphate: identification of two peptides from the ATP-binding domain

1 reference

12 December 2020

Surface modification of magnetic nanoparticle via Cu(I)-catalyzed alkyne-azide [2 + 3] cycloaddition

1 reference

12 December 2020

Toward selective histone deacetylase inhibitor design: homology modeling, docking studies, and molecular dynamics simulations of human class I histone deacetylases

1 reference

12 December 2020

Identifiers

DOI

10.1021/JM9005077

1 reference

20 August 2017

1 reference

20 August 2017

PubMed publication ID

19886628

1 reference