Synthesis and structure-activity relationships of antimalarial 4-oxo-3-carboxyl quinolones. (Q39627889)

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19 January 2020

title

Synthesis and structure-activity relationships of antimalarial 4-oxo-3-carboxyl quinolones (English)

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19 January 2020

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7

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2

W Armand Guiguemde

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Michele C Connelly

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4

Fangyi Zhu

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3

Martina Sigal

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Solomon Nwaka

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19 January 2020

author name string

Yiqun Zhang

series ordinal

1

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language of work or name

English

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publication date

11 February 2010

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Bioorganic & Medicinal Chemistry

19 January 2020

published in

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volume

18

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issue

7

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19 January 2020

page(s)

2756-2766

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Enhancement of the antimalarial activity of ciprofloxacin using a double prodrug/bioorganometallic approach

19 January 2020

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14 September 2017

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Induction of calf thymus topoisomerase II-mediated DNA breakage by the antibacterial isothiazoloquinolones A-65281 and A-65282

14 September 2017

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14 September 2017

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15 June 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/20206533

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Mammalian topoisomerase II inhibitory activity of 1-cyclopropyl-6,8- difluoro-1,4-dihydro-7-(2,6-dimethyl-4-pyridinyl)-4-oxo-3-quinolinecarb oxylic acid and related derivatives

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20206533

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BMC.2010.02.013

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20206533%20AND%20SRC:MED&resulttype=core&format=json

19 January 2020

1 reference

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19 January 2020

PubMed publication ID

20206533

1 reference