Discovery of potent and selective histone deacetylase inhibitors via focused combinatorial libraries of cyclic alpha3beta-tetrapeptides (Q33496543)

27 July 2017

title

Discovery of potent and selective histone deacetylase inhibitors via focused combinatorial libraries of cyclic alpha3beta-tetrapeptides (English)

1 reference

27 July 2017

Christian A Olsen

1

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author name string

M Reza Ghadiri

series ordinal

2

1 reference

27 July 2017

language of work or name

English

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publication date

1 December 2009

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Journal of Medicinal Chemistry

27 July 2017

published in

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27 July 2017

volume

52

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27 July 2017

issue

23

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27 July 2017

page(s)

7836-7846

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Probing the bioactive conformation of an archetypal natural product HDAC inhibitor with conformationally homogeneous triazole-modified cyclic tetrapeptides.

27 July 2017

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21 June 2018

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12 December 2020

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Design and Synthesis of Cyclopeptide Analogues of the Potent Histone Deacetylase Inhibitor FR235222

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12 December 2020

Identifiers

DOI

10.1021/JM900850T

1 reference

27 July 2017

1 reference

27 July 2017

1 reference