The effect of conformation on the membrane permeation of coumarinic acid- and phenylpropionic acid-based cyclic prodrugs of opioid peptides. (Q44352355)

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10 December 2019

title

The effect of conformation on the membrane permeation of coumarinic acid- and phenylpropionic acid-based cyclic prodrugs of opioid peptides (English)

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10 December 2019

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3

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10 December 2019

Binghe Wang

5

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10 December 2019

author name string

O S Gudmundsson

1

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10 December 2019

S D Jois

2

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10 December 2019

T J Siahaan

4

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10 December 2019

R T Borchardt

6

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10 December 2019

publication date

1 April 1999

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Chemical Biology and Drug Design

10 December 2019

published in

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10 December 2019

volume

53

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10 December 2019

issue

4

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10 December 2019

page(s)

383-392

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Recent developments in the design of receptor specific opioid peptides

10 December 2019

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Synthesis and evaluation of the physicochemical properties of esterase-sensitive cyclic prodrugs of opioid peptides using coumarinic acid and phenylpropionic acid linkers

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Coumarinic acid-based cyclic prodrugs of opioid peptides that exhibit metabolic stability to peptidases and excellent cellular permeability

21 January 2018

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Phenylpropionic acid-based cyclic prodrugs of opioid peptides that exhibit metabolic stability to peptidases and excellent cellular permeation

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How structural features influence the biomembrane permeability of peptides

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Transferred nuclear Overhauser effect analyses of membrane-bound enkephalin analogues by 1H nuclear magnetic resonance: correlation between activities and membrane-bound conformations

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The effect of beta-turn structure on the permeation of peptides across monolayers of bovine brain microvessel endothelial cells

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Effect of stereochemistry on the transport of Aca-linked beta-turn peptidomimetics across a human intestinal cell line

21 January 2018

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Acyloxyalkoxy-based cyclic prodrugs of opioid peptides: evaluation of the chemical and enzymatic stability as well as their transport properties across Caco-2 cell monolayers

21 January 2018

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The effect of conformation of the acyloxyalkoxy-based cyclic prodrugs of opioid peptides on their membrane permeability

21 January 2018

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Prodrug strategies to enhance the intestinal absorption of peptides

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Novel esterase-sensitive cyclic prodrugs of a model hexapeptide having enhanced membrane permeability and enzymatic stability

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Synthesis of a Novel Esterase-Sensitive Cyclic Prodrug System for Peptides That Utilizes a “Trimethyl Lock”-Facilitated Lactonization Reaction

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Coumarin-based prodrugs 2. Synthesis and bioreversibility studies of an esterase-sensitive cyclic prodrug of dadle, an opioid peptide

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21 January 2018

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7 January 2021

Synthesis and biological properties of gamma-glutamyl-dermorphin, a prodrug

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7 January 2021

The effect of conformation on membrane permeability of an acyloxyalkoxy-linked cyclic prodrug of a model hexapeptide

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7 January 2021

Esterase-sensitive cyclic prodrugs of peptides: evaluation of an acyloxyalkoxy promoiety in a model hexapeptide

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7 January 2021

Effect of restricted conformational flexibility on the permeation of model hexapeptides across Caco-2 cell monolayers

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7 January 2021

The effect of beta-turn structure on the passive diffusion of peptides across Caco-2 cell monolayers

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7 January 2021